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“像在市医院,也是没有条件更没有想起要样做的。”胡岱源补充说。

“嗯,做得好!”禹若冰夸完后,开口问道:“你打电话说,有重要的发现,究竟是怎么回事?”

“嗨,这事说来可就话长了。金副所长,这事儿还是你来汇报吧。”胡岱源说道。

“胡主任,你掌握的全面一些,还是您汇报更好一些。”在市医院的时候,胡岱源毕竟是金兆铭的上级,来到集团的科研所,他的排名虽说在金兆铭之后,小金大夫还是挺尊重他的。

“别推三阻四的了,胡所长,我和金所长实际上来科研所的时间不长,具体还是由你向集团领导汇报吧。”孟先德一语定音。

“好吧。在市医院时,我们虽然从食肉植物提炼出能攻破病毒外壳保护层的蛋白酶,但是屡次试验发现,它们的活性有些差攻击力并不强。”胡岱源说:“这状况有点儿像有些运动员,在赛场缺乏活力,所以就有人背地里服用兴奋剂……”

“什么?你是说,中草药也有兴奋剂?”几个人异口同声地嚷出来。

不过,事实也的确如此。”胡岱源不紧不慢地说道:“赵老在分析我们的研究成果时,就曾经批评说,我们只关注了中医经方中的君臣辅佐,而忽略了即使是同一味中药,也有君臣成分存在。孟所和金所履职后,我们一起研讨赵老的见解,金副所长从微生物药动力学的现代研究成果中,给我们一个启示:我们所提取的两种蛋白质分解酶,还缺乏类似‘兴奋剂’那样的‘刺激’,真地需要加以激活!至于究竟是怎么回事,接下来,请小金先就这个发现补充汇报吧。”

禹若冰晓得,金兆铭在省中医药大学读的研究生课题,就是中药动力学这个冷门的。便把目光投向他。

“这种状况的出现,恐怕还得多啰嗦几句,要从中西药的根本区别说起。”金兆铭轻轻咳嗽一声,在组织语言后才说道:“中药和西药最大的区别就在于分子结构不同。一般说来,西药大都是具有靶向性的单分子和小分子结构,就像对敌作战中的制导导弹或火箭炮那档的重武器,对着敌方倒是能够准确加以打击,所以人们普遍认为西药见效快。然而,西药最大的弊端,就是攻其一点不及其余。在狂轰滥炸中,顽敌虽然被消灭,但是往往波及无辜,甚至伤及无辜,造成人体内的正常细胞乃至器官的损伤。这就是西药往往难以避免的‘副作用’。我们如果认真地审读那些西药的《药品说明书》,几乎都有‘副作用’这一栏的说明。”

说到这里,他稍微一顿,话题一转继续说道:“中药除了矿物类之外,绝大多数是多种分子团和高分子有机化合物结构,并非像西药那样的单一成分、单一效应。举个最常见的例子,当归是一种典型的常见中药材,但是当归头可补血和止血,当归身或全株既可补血,亦有养血之效,当归尾单用却破血扫血。同一味药,却能对症治疗多种病症。西药可就没这么好使了。”

“话题扯远了吧?你直接向领导说发现了什么。”胡岱源插嘴打断说。

“哦,对不起,有点儿扯远了。”金兆铭不好意思地说道,把话头扯回正题:“我们在探讨从中草药中提取的蛋白质分解酶为什么效用不好时,正好看到相关的论文,认为各种酶只有在最适的温度范围内,酶的活性才最强,酶促反应的速度最大。据科学实验,在适宜的温度范围内,温度每升高十摄氏度,酶促反应速度可以相应提高一至两倍。而且,不同生物体内酶的最适温度也不同,例如动物组织中各种酶的最适温度为三十七至四十摄氏度,而微生物体内各种酶的最适温度为二十五至六十摄氏度。”

“这和你们的什么发现有什么直接关联?”秦苏怡的眉头微皱,插嘴问道。

“如果环境温度的条件达不到,那么就应当想方设法把酶的活性激发出来。这就是胡主任刚才譬喻的运动员的‘兴奋剂’,那玩意儿在体育界是绝对禁用的,但是对于我们的科研来说,却是必须找到的!”金兆铭的话,逐渐接近了“谜团”的揭开:“能激活酶的物质称为酶的激活剂。目前已经被发现的激活剂的种类很多,包括无机阳离子,如钠离子、钾离子、铜离子、钙离子等;无机阴离子,如氯离子、溴离子、碘离子、硫酸盐离子、磷酸盐离子等;有机化合物,如维生素C、半胱氨酸等。”金兆铭一口气说出了一连串的名字后,解释说:“许多酶的活性状态差的时候,必须经过适当的激活剂激活后才具有活性。”

“你的意思是说, 咱们千辛万苦提取的那两种蛋白质分解酶,还需要找到它们的激活剂才能物尽其用。这又到哪里去找?”秦苏怡的眉头越趋越紧,喃喃说道。

“那倒不用发愁。正如赵老爷子所言,单就某一味中草药来说,其药性也有君臣之分。我据此分析,前一阵子提取蛋白质分解酶时,恰恰忽视了这一点,只提取了分解酶这一‘君药’组分,而忽略了其中的‘臣药’组分,所以才导致它们攻破病毒防护层的能力衰减,发挥不了全力的作用……”孟先德说道。

“从我们在赵老指导下对《端木医案》的研究分析,把端木大夫在医治蛇缠腰时所用的各种药材疏理了一遍,认为分解酶的激活剂也有可能存在于其中,于是重开实验……”胡岱源接着说道:“基于这一新的认识,我们像过筛子般进行了几百次实验。幸亏药厂移交过来的实验仪器和检测设备足够多,而且从药厂过来的实验员个顶个的是业务高手, 并且有电子显微镜‘坐镇中帐’,很快就见成果。唉如果还是在医院做,还不晓得要搞到猴年马月哩!”

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